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Epinastine HCl
CAS No. 108929-04-0
Epinastine HCl ( Epinastine Hydrochloride | Alesion | Elestat )
产品货号. M17804 CAS No. 108929-04-0
Epinastine 是一种抗组胺剂和肥大细胞稳定剂，用于治疗过敏性结膜炎的滴眼剂。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 25MG | ￥405 | 有现货 |
|
| 50MG | ￥527 | 有现货 |
|
| 100MG | ￥786 | 有现货 |
|
| 200MG | ￥1482 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Epinastine HCl
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Epinastine 是一种抗组胺剂和肥大细胞稳定剂，用于治疗过敏性结膜炎的滴眼剂。
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产品描述Epinastine Hydrochloride is a histamine H1 receptor antagonist without sedative activity. Epinastine hydrochloride blocks the histamine H1 receptor and inhibits the release of histamine from mast cells. This prevents the typical allergic symptoms that are caused by histamine activity on capillaries, skin, and mucous membranes. Typical histamine activities include vasodilation, bronchoconstriction, increased vascular permeability, pain, itching, and spasmodic contractions of gastrointestinal smooth muscles. Epinastine HCl also has affinity for histamine H2, 5-HT2, and the alpha-1, alpha-2 adrenergic receptors.
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体外实验——
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体内实验——
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同义词Epinastine Hydrochloride | Alesion | Elestat
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通路Others
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靶点Other Targets
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受体HT
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研究领域Inflammation/Immunology
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适应症——
化学信息
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CAS Number108929-04-0
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分子量285.77
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分子式C16H15N3·HCl
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纯度>98% (HPLC)
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溶解度In Vitro:?H2O : 100 mg/mL (349.93 mM)
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SMILESCl[H].NC1=NCC2N1C1=CC=CC=C1CC1=CC=CC=C21
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化学全称3-Amino-9,13b-dihydro-1H-dibenzo[c,f]imidazo[1,5-a]azepine Hydrochloride
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Fügner A, et al. Arzneimittelforschung, 1988, 38(10), 1446-1453.
产品手册
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